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¥­¡¼¥ï¡¼¥É:inhibitor ¤Î¸¡º÷·ë²Ì

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2C2a11
2024/03/25 11:36
C2
Isolation, structure elucidation, and biological activities of sesquiterpenes and phthalides from two edible mushrooms Pleurotus species
¡ûJewel De Padua1, Emi Fukushima Sakuno2, Kotomi Ueno3, Thomas Edison dela Cruz4, Atsushi Ishihara3
1The United Graduate School of Agricultural Sciences, Tottori University, Tottori, Japan, 2The Tottori Mycological Institute, The Japan Kinoko Research Center Foundation, Tottori, Japan, 3Faculty of Agriculture, Tottori University, Tottori, Japan, 4Department of Biological Sciences, College of Science, University of Santo Tomas, Espa¢®a Blvd., Manila, Philippines
2C3a09
2024/03/25 11:06
C3
ÅìÆ¥¸¥¢¸¶»º¥ê¥°¥Î¥»¥ë¥í¡¼¥¹·Ï¥Ð¥¤¥ª¥Þ¥¹¤ò¸¶ÎÁ¤È¤·¤¿PHBÀ¸»º
PHB production from lignocellulosic biomass native to Southeast Asia
¡û¹Ó°æ δ±×1¡¢ÍõÀî ¿¸Ê¿1¡¢Sudesh Kumar2¡¢Fazita MR Nurul2¡¢Cheu Peng Leh2¡¢Haafiz MK Mohamad2¡¢Guan Seng Tay2¡¢¾®¿ù ¾¼É§1
¡ûTakamitsu Arai1, Shimpei Aikawa1, Kumar Sudesh2, Nurul Fazita MR2, Leh Cheu Peng2, Mohamad Haafiz MK2, Tay Guan Seng2, Akihiko Kosugi1
1¹ñºÝÇÀ¸¦¡¢2¥Þ¥ì¡¼¥·¥¢Íý²ÊÂç
1Japan International Research Center for Agricultural Sciences, 2School of Biological Sciences, Universiti Sain Malaysia
2C4p12
2024/03/25 16:07
C4
¶â°°Í¸À­¥×¥í¥Æ¥¤¥ó Ser/Thr ¥Û¥¹¥Õ¥¡¥¿¡¼¥¼ 1A¿·µ¬Á˳²ºÞ¤ÎÁ˳²µ¡¹½²òÀÏ
Identification and characterization of novel inhibitors of metal-dependent protein Ser/Thr phosphatase 1A
¡ûÎëÌÚ ·òͧ1¡¢¾®Åç ½ÙÌé2¡¢ñÁ¼ ½¤2¡¢ÂçÀ¾ ÁÇ»Ò1
¡ûTaketomo SUZUKI1, Syunya KOJIMA2, Osamu NIYOMURA2, Motoko OHNISHI1
1ÃæÉôÂ籡±þÀ¸¡¢2ÃæÉôÂç±þ²½
1Graduate School of Bioscience and Biotechnology, Chubu Univ., 2Department of Applied Chemistry, Chubu Univ.
2C4p13
2024/03/25 16:18
C4
3,5-¥¸¥¬¥í¥¤¥ë¥Õ¥é¥Ð¥ó-3-¥ª¡¼¥ëͶƳÂΤÎ3°Ì¤ÎΩÂΤ¬³èÀ­¤ä¥¿¥ó¥Ñ¥¯¼Á¤È¤ÎÁê¸ßºîÍѤËÍ¿¤¨¤ë±Æ¶Á
Effect of the 3-position of 3,5-digalloylflavan-3-ol derivatives on their activity and interaction with proteins
¡ûËÙ¸ý ÎÊÂÀ1¡¢ÀÄÌÚ ´Ä1¡¢Æ»²¼ ν1¡¢¼¼°æ À¿3¡¢Ä¹ÅÄ ÍµÇ·3,4¡¢óîÆ£ °Âµ®»Ò1,2
¡ûRyouta Horiguchi1, Atoru Aoki1, Ryo Doge1, Makoto Muroi3, Hiroyuki Osada3,4, Akiko Saito1,2
1ÂçºåÅÅÄÌÂ籡¹©¡¢2ÂçºåÅÅÄÌÂ繩¡¢3Íý¸¦CSRS¡¢4ÀŲ¬¸©Î©ÂçÌô
1Graduate School of Engineering, OECU, 2Department of Environmental Science, Faculty of Engineering, OECU, 3RIKEN Center for Sustainable Resource Science, 4Division of Pharmaceutical Sciences, School of Pharmaceutical Sciences, University of Shizuoka
2C5p11
2024/03/25 15:56
C5
ÈùÀ¸Êª¤ËÂФ¹¤ë¶õµ¤¥Õ¥¡¥¤¥ó¥Ð¥Ö¥ë¤Î¸ú²Ì¤Ë´Ø¤¹¤ëÄ´ºº
Investigation of the effect of air-fine bubbles on microorganisms
¡û´äºê ¤Ê¤Ä¤Í1¡¢Ë­ÅÄ ·òÂÀ1¡¢Æ²ËÜ ¼Âºé´õ1¡¢Â¿ÅÄ ²Â¿¥2¡¢À¾Æâ ͪʹ2¡¢Â§Â¼ »ËÊâ1¡¢¿Á δ»Ö2¡¢À¾ËÜ ¿¿¶×1
¡ûNatsune IWASAKI1, Kenta TOYODA1, Misaki DOMOTO1, Kaori TADA2, Yusuke NISHIUTI2, Shiho NONORIMURA1, Takashi HATA2, Makoto NISHIMOTO1
1ϹâÀì¡¢2¹âÃιâÀì
1NIT, Wakayama College, 2NIT, Kochi College
2D2a01
2024/03/25 09:30
D2
¿©Éʲù©¾ò·ï¤ª¤è¤Ó°ßIJ¾Ã²½¤Ë¤ª¤±¤ë¿©ÍÑÁôÎàͳÍè¤ÎDPP-4Á˳²¥Ú¥×¥Á¥É¤Î°ÂÄêÀ­
Stability of DPP-4 inhibitory peptides from edible algae under food processing conditions and gastrointestinal digestions
¡ûåéÈ· ¹¯ÂÀ¡¢º´Æ£ ºÚ±û¡¢ÈÓÅç ÍÛ»Ò¡¢¿ù»³ ·òÆóϺ
¡ûKota Ebato, Nao Sato, Yoko Iijima, Kenjiro Sugiyama
¹©³Ø±¡Âç
The Univ. of Kogakuin
2D4p12
2024/03/25 16:07
D4
¥Û¥ë¥â¥óÀ©¸æºÞNJ15¤Î¿¢ÊªÉ½ÁؤËÍ¿¤¨¤ë±Æ¶Á¤Î²òÀÏ
Analysis of the effects of the phytohormone signal transduction inhibitor NJ15 on plant surface layers
¡ûºä¾å ÆࡹÈÁ¡¢ÃæÅè ÀµÉÒ¡¢Àõ¸« ÃéÃË
¡ûNanaho SAKAUE, Masatoshi NAKAJIMA, Tadao ASAMI
ÅìÂ籡¡¦ÇÀÀ¸²Ê
The Univ. of Tokyo
2D7p07
2024/03/25 15:04
D7
¥¤¥ÍͳÍ迵¡Ç½À­¥Ú¥×¥Á¥É¤Îµ¡Ç½À­¸þ¾å¤Ë´Ø¤¹¤ë¸¦µæ
Studies on functional improvement of multifunctional peptide from rice
¡û±óÆ£ ¤á¤¤1¡¢Å쳤ÎÓ ÍµæÆ1¡¢ÎëÌÚ Í¥Èô1¡¢Ã«¸ý ÀµÇ·2¡¢ÅÄÃæ ¹§ÌÀ1¡¢Íî¹ç ½©¿Í1
¡ûMei ENDO1, Hiroto TOKAIRIN1, Yuhi SUZUKI1, Masayuki TANIGUCHI2, Takaaki TANAKA1, Akihito OCHIAI1
1¿·³ãÂ籡¼«Á³¸¦¡¢2¿·³ãÀÄÎÍûÂ硦¿Í´ÖÁí¹ç
1Grad. Sch. of Sci. Technol., Niigata Univ., 2Dep. of Liv. Stu., Niigata Seiryo Jnr. Col.
2E5a01
2024/03/25 09:30
E5
ÈùÀ¸Êª¤òÍøÍѤ·¤¿½ÏÀ®¥µ¡¼¥â¥ó¤Ë´Þ¤Þ¤ì¤ë·ì°µ¹ß²¼ºîÍÑʪ¼Á¤ÎʬÀÏ
Analysis of substances with hypotensive effects from salmon aged with microorganisms
¡ûÊÒ»³ ÂÀÃÒ1¡¢Â¼¾å ¼þ°ìϺ2
¡ûTaichi KATAYAMA1, Shuichiro MURAKAMI2
1ÌÀÂ籡ÇÀ¡¢2ÌÀÂçÇÀ
1Meiji Univ. School of Agriculture, 2Meiji Univ.
3C2a01
2024/03/26 09:30
C2
¿·µ¬¥Ú¥×¥Á¥É¥°¥ê¥«¥óÀ¸¹çÀ®·ÐÏ©Á˳²ºÞ¤Îõº÷
Searching for Specific Inhibitors of the Alternative Peptidoglycan Biosynthetic Pathway
ÇßÄÅ ½¨Ê¿1¡¢³ÑÅÄ µ£2¡¢µ´Ìø ½Õ²Ö1¡¢°ð¶¶ ͤµ¯3,4¡¢ÌîÃæ ·ò°ì3,4¡¢¡û¾®³Þ¸¶ ÂÙ»Ö2¡¢ÂçÍø Å°2
Shuhei UMETSU1, Takeshi TSUNODA2, Haruka KIYANAGI1, Yuki INAHASHI3,4, Kenichi NONAKA3,4, ¡ûYasushi OGASAWARA2, Tohru DAIRI2
1ËÌÂ籡Áí²½¡¢2ËÌÂ籡¹©¡¢3ËÌΤÂçÂ缸¦¡¢4ËÌΤÂ籡´¶À÷À©¸æ
1Grad. Sch. Chem. Sci. Eng., Hokkaido Univ., 2Grad. Sch. Eng., Hokkaido Univ., 3Omura Inst., Kitasato Univ., 4Grad. Sch. Infection Cont., Kitasato Univ
3C2a02
2024/03/26 09:41
C2
¿·µ¬¥á¥Ê¥­¥Î¥óÀ¸¹çÀ®·ÐÏ©Á˳²ºÞ¤Îõº÷
Searching for Specific Inhibitors of the Alternative Menaquinone Biosynthetic Pathway
¡ûµ´Ìø ½Õ²Ö1¡¢µÆÃÓ ËãΤ¹¾1¡¢³ÑÅÄ µ£2¡¢ÌîÃæ ·ò°ì3,4¡¢°ð¶¶ ͤµ¯3,4¡¢¾®³Þ¸¶ ÂÙ»Ö2¡¢ÂçÍø Å°2
¡ûHaruka KIYANAGI1, Marie KIKUCHI1, Takeshi TSUNODA2, Kenichi NONAKA3,4, Yuki INAHASHI3,4, Yasushi OGASAWARA2, Tohru DAIRI2
1ËÌÂ籡Áí²½¡¢2ËÌÂ籡¹©¡¢3ËÌΤÂçÂ缸¦¡¢4ËÌΤÂ籡´¶À÷À©¸æ
1Grad. Sch. Chem. Sci. Eng., Hokkaido Univ., 2Grad. Sch. Eng., Hokkaido Univ., 3Omura Inst., Kitasato Univ., 4Grad. Sch. Infection Cont., Kitasato Univ
3C4p02
2024/03/26 14:01
C4
11¦Â-HSD1¤òÁ˳²¤¹¤ë¥á¥í¥Æ¥ë¥Ú¥Î¥¤¥É¤Î¹çÀ®¸¦µæ
Synthetic study of meroterpenoids as 11¦Â-HSD1 inhibitor
¡û²ÃÆ£ ¸÷µ±¡¢¹â¶¶ À²ÂÀϺ¡¢¾¡ÅÄ Î¼¡¢ÀпÀ ·ò¡¢¼ã¿¹ ¿¸Ç·²ð
¡ûMitsuki KATO, Seitaro TAKAHASHI, Ryo KATSUTA, Ken ISHIGAMI, Shinnosuke WAKAMORI
ÅìÇÀÂ硦À¸Ì¿
Tokyo Univ. of Agriculture
3C4p08
2024/03/26 15:15
C4
¥ß¥È¥³¥ó¥É¥ê¥¢µ¡Ç½Á˳²ºÞfusaramin¤ÎÁ´¹çÀ®¤Ë¤è¤ëΩÂβ½³Ø¹½Â¤¤Î·èÄê¡¢¹½Â¤³èÀ­Áê´Ø¤Î²òÌÀ¡¢¿·µ¬¹³¿¿¶Ý³èÀ­¤Îȯ¸«
Determination of the Stereochemical Structure, Elucidation of the Structure-Activity Relationship, and the Discovery of Novel Antifungal Activities by the Total Synthesis of Fusaramin, an Inhibitor of Mitochondrial Function
¡û·¯Åè °ª1,2¡¢ÇëËÜ ÂçÃÏ1¡¢Ëܾ± ²í»Ò1,2¡¢ºä°æ ¹î¹Ô1¡¢ËÜ´Ö ñ¥ÂÀ1,2¡¢Æ£ ¿¸°ì3¡¢´ä·î Àµ¿Í1,2¡¢¾ïÈ× ½ÓÇ·2¡¢ÌîÃæ ·ò°ì1,2¡¢ÃÎÇ° Âó¼Â4¡¢±±°æ ·òϺ5¡¢Àõ¸« ¹Ô¹°1,2
¡ûAoi Kimishima1,2, Daichi Hagimoto1, Masako Honsho1,2, Katsuyuki Sakai1, Sota Honma1,2, Shin-ichi Fuji3, Masato Iwatsuki1,2, Toshiyuki Tokiwa2, Kenichi Nonaka1,2, Takumi Chinen4, Takeo Usui5, Yukihiro Asami1,2
1ËÌΤÂ籡´¶À÷À©¸æ¡¢2ËÌΤÂçÂ缸¦¡¢3½©Åĸ©ÂçÀ¸»ñ¡¢4ÅìÂ籡Ìô¡¢5ÃÞÇÈÂçÀ¸Ì¿´Ä¶­
1Kitasato University, 2Ōmura Satoshi Memorial Institute, 3Akita Prefectural University, 4The Univ. of Tokyo, 5University of Tsukuba
3C7a06
2024/03/26 10:33
C7
Æî¶Ë¥æ¥­¥É¥ê±ÄÁãÀפ«¤éʬΥ¤·¤¿ÈùÀ¸Êª¤«¤é¤Î¥Ð¥¤¥ª¥Õ¥£¥ë¥àÁ˳²Êª¼Á¤Î¥¹¥¯¥ê¡¼¥Ë¥ó¥°
Screening for biofilm inhibitors from microorganisms isolated from Antarctic snow petrel nesting sites
¡û°¤ºÂ¾å ¹°¹Ô1,2¡¢ÌÚ²¼ ñ¥1¡¢SIDDIQA Ayesha1¡¢ÎÓ ¾»Ê¿3
¡ûHiroyuki AZAKAMI1,2, Hayato KINOSHITA1, Ayesha SIDDIQA1, Shohei HAYASHI3
1»³¸ýÂçÇÀ¡¢2»³¸ýÂçÃæ¹â²¹Èù¥»¡¢3Å纬ÂçÀ¸Êª»ñ¸»
1Fac. of Agr., Yamaguchi Univ, 2RCTMR, Yamaguchi Univ, 3Fac. of Life Env. Sci., Simane Univ.
3C7a14
2024/03/26 12:09
C7
Æó¼¡Âå¼ÕʪÀ¸¹çÀ®¹ÚÁÇÁ˳²ºÞ¤òÍѤ¤¤¿¿·µ¬²½¹çʪ¤Îõº÷·Ï¤Î¹½ÃÛ
Establishment of natural product screening system using biosynthetic enzyme inhibitor
üâ¼ °ê¼Â1¡¢ÌîÀî ½Óɧ2¡¢²¬Ìî °¡µª»Ò2¡¢±ÛÌî ¹­Àã2¡¢¾ÂËÜ Êæ1¡¢ÏÂÅÄ Âç1¡¢¡û²ÃÆ£ ľ¼ù1
Ikumi TAKAMURA1, Toshihiko NOGAWA2, Akiko OKANO2, Hiroyuki KOSHINO2, Minori NUMAMOTO1, Masaru WADA1, ¡ûNaoki KATO1
1ÀÝÆîÂ硦ÇÀ¡¢2Íý¸¦CSRS
1Setsunan Univ., 2RIKEN CSRS
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